What is Varenicline tartrate?

Varenicline tartrate powder, also known as tartrate swab. Its chemical name is(- tetrahydro-2-methyl-3-( 3- pyridyl) -1,5-benzodiazepin-7-yl)( 1,4- dihydroxy) dipyrophosphate. It's a white to out-white crystalline powder， it's answerable in water and methanol at room temperature. its molecular formula isC13H13N3.C4H6O6P2, its relative molecular mass is361.3 g/ spook, CAS number is 375815-87-5. Its pharmacological medium of action involves binding to α4β2 nicotinic acetylcholine receptors on neurons, cranking these receptors, and adding dopamine release, producing nicotine- suchlike goods. it can reduce tobacco dependence in smokers by mimicking the goods of nicotine while reducing pullout symptoms associated with quitting smoking. its development began in the late 1990s when Pfizer invested heavily to find a more effective smoking conclusion drug. Their exploration concentrated on nicotinic receptors, hoping to develop a medicine that could mimic nicotine's goods and reduce pullout symptoms.

 After expansive trial and testing, experimenters successfully synthesized Varenicline tartrate API. The medicine was approved by the US FDA in 2006 and latterly approved for use in numerous countries. Since its blessing, it has been shown to be a largely effective smoking conclusion drug, significantly reducing tobacco dependence and easing pullout symptoms. Despite some contestation and reports of adverse events, it remains a favored choice for numerous who wish to quit smoking. Overall, the development of Varenicline tartrate involved times of exploration and development, eventually achieving tremendous success and getting an important treatment for smoking conclusion.

Basic Information

Quality standard

Stability & Storage

Varenicline tartrate powder is relatively stable, but under certain conditions, it may undergo degradation or decomposition. Its stability can be described as follows:

Thermal stability it's fairly stable at room temperature, but it can suffer partial declination under high temperature and moisture conditions. At 60 °C, it has good stability, and after being stored at room temperature for 24 months, its quality remains above 98.

Light stability it's fairly stable to light, but it gradationally loses exertion when exposed to strong light and ultraviolet radiation. thus, it should be defended from exposure to strong light and ultraviolet radiation during product and storehouse.

Oxidative stability it has good oxidation stability, it may be degraded if exposed to egregious oxidants( similar as hydrogen peroxide and Potassium permanganate).

Acid- alkali stability it's sensitive to the acid- alkali terrain, and storing it in an acidic or alkaline terrain may lead to declination.

In summary, to insure the quality and stability, it should be defended from exposure to high temperature, light, oxidants, and acidic or alkaline surroundings. Applicable storehouse conditions, similar as blankness, low light, and low temperature, should be used. When using the medicine, attention should also be paid to its quality and expiration date to avoid affecting its efficacity.

Storage requirements

Storage temperature: VareniclineTartrate should be stored in a dry, cool, and well-ventilated place, with the optimal temperature range being 2°C-8°C. Storing it at this temperature can maintain the quality and stability of the drug and extend its shelf life.

Light protection: it is sensitive to light, so opaque containers should be used to protect the drug during storage to avoid direct sunlight or strong light exposure. Avoid exposure to UV lamps.

Moisture-proof: it is hygroscopic, so moisture should be avoided during storage. Sealed packaging and bioreagent desiccants can be used to prevent moisture from entering.

No freezing: it is not resistant to freezing and cannot be stored or transported under frozen conditions, otherwise it will cause drug degradation and loss of efficacy.

Avoid vibration: it is a powder, and if it undergoes vibration or shock during storage or transportation, it may break or deform, affecting its quality and activity.

In summary, to protect the quality and stability,it should be followed during storage and transportation. Particularly, factors such as temperature, light, humidity, and vibration, once exceeding the tolerance range of the drug, would lead to drug failure or degradation.

Packing & Shipping

Packing: 1kg/foil bag;5kg/carton;25kg/fiber drum; or packing as your request.

Customization: Customized logo; Customized packaging; Graphic customization

Shipping:

Payment Term

Why Choose Xi'an Yihui?

Customer feedback

Xi'an Yihui certificates

Xi'an Yihui Factory & Warehouse

Our Advantage

Rich experience: we have 13 Years of professional experience;

Customers all over the world: sell to more than 100 countries;

Provide diversified products: the products have been applied to all major international brands in the fields of drugs, dietary supplements, cosmetics, animal nutrition and functional food.

Price advance: low MOQ with competitive price;

Quality certification: ISO; Halal; Kosher certified

After-sales service: Professional team 7*24 hours customer service.

In conclusion

In summary, Xi'an Yihui company as a professional Varenicline Tartrate powder manufacturer, has strong technical strength and advanced production equipment and is committed to providing customers with high-quality, efficient, and reliable drug raw materials. if you need it, pls feel free to contact us any time. we will reply you asap.

Our contact information:

E-mail: sales@yihuipharm.com
Tel: 0086-29-89695240
WeChat or WhatsApp: 0086-17792415937

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